The drug atlas
Child Health/Paediatric antiepileptics & status

Seizures & status epilepticus (paeds)

also: buccal midazolam · status epilepticus · sodium valproate · ethosuximide · AED

Overview

The status-epilepticus escalation ladder plus the maintenance antiepileptics by seizure type. The valproate teratogenicity restriction and the absence-seizure choice are heavily tested.

Mechanism

Benzodiazepines enhance GABA-A inhibition (abort seizures). Sodium valproate broadens inhibition (↑GABA, Na-channel) — broad spectrum. Ethosuximide blocks T-type calcium channels in thalamic neurones (absence). Carbamazepine/lamotrigine/phenytoin stabilise voltage-gated Na channels (focal/GTC).

Indications

  • Status epilepticus (emergency)
  • Maintenance therapy for epilepsy by seizure type
  • Febrile convulsions (usually no regular treatment)

The agents

Buccal midazolam / PR diazepamcommunity 1st step

First benzodiazepine dose (home/ambulance).

IV lorazepamhospital 1st step

repeat once after 10 min

In-hospital benzodiazepine.

IV phenytoin / levetiracetam2nd line (status)

If 2 benzo doses fail → call for help, prep for ICU/thiopental.

Sodium valproateGTC/myoclonic

Broad-spectrum but TERATOGENIC — avoid in girls/women of childbearing potential (pregnancy prevention programme).

Ethosuximideabsence

First-line for absence seizures.

Carbamazepine / lamotriginefocal

Carbamazepine can WORSEN absence/myoclonic seizures.

Adverse effects

Valproate: teratogenicity (neural tube defects)serious

Plus weight gain, tremor, hepatotoxicity, hair loss, pancreatitis.

Carbamazepine: SJS, hyponatraemia (SIADH), enzyme inductionserious
Phenytoin: gum hypertrophy, ataxia, zero-order kineticscommon
Lamotrigine: Stevens-Johnson syndrome (slow titration)serious
Benzodiazepines: respiratory depressionserious

Cautions & contraindications

Sodium valproate in girls / women of childbearing potentialpaediatric

Teratogen — only under a pregnancy prevention programme when no alternative.

Carbamazepine in absence/myoclonic epilepsyall

Can exacerbate them.

Interactions

  • Carbamazepine/phenytoin induce CYP (↓OCP, ↓other AEDs)
  • Valproate inhibits lamotrigine metabolism (↑SJS risk)

Monitoring & kinetics

Status: ABC, glucose, timing; phenytoin levels/ECG,Valproate: LFTs; pregnancy prevention

Status ladder: benzo → repeat benzo → phenytoin/levetiracetam → RSI/thiopental + ICU. Do not stop AEDs abruptly.

Source: NICE NG217 — Epilepsies · APLS — Status epilepticus