The drug atlas
Cardiovascular/Antiarrhythmic (Vaughan-Williams)

Antiarrhythmics (adenosine, flecainide, lidocaine)

also: adenosine · flecainide · lidocaine · Vaughan-Williams · SVT

Overview

The antiarrhythmics not covered by the rate-control cards — adenosine for SVT, flecainide for paroxysmal AF, lidocaine for VT — organised by the Vaughan-Williams classification.

Mechanism

Vaughan-Williams: I = Na-channel blockers (Ia procainamide, Ib lidocaine, Ic flecainide); II = β-blockers; III = K-channel blockers (amiodarone, sotalol); IV = non-DHP CCBs. Adenosine is unclassified — transiently blocks the AV node (A1 receptor → ↑K⁺ efflux, hyperpolarisation) → breaks AV-nodal re-entry SVT.

Indications

  • SVT (adenosine — diagnostic + therapeutic)
  • Paroxysmal AF / "pill-in-the-pocket" (flecainide)
  • Ventricular tachycardia (lidocaine/amiodarone)

The agents

AdenosineAV-node block (SVT)

rapid IV bolus 6→12→18 mg

Transient flushing/chest tightness/"sense of doom"; very short t½. CI in ASTHMA → use verapamil. Give via a large vein, fast, with a flush.

FlecainideClass Ic

oral / "pill-in-pocket"

Paroxysmal AF in structurally normal hearts; AVOID post-MI / structural/ischaemic heart disease (pro-arrhythmic).

LidocaineClass Ib

IV

Ventricular arrhythmias; also a local anaesthetic.

ProcainamideClass Ia

IV

VT, and AF in WPW pre-excitation.

Adverse effects

Adenosine: transient asystole/bradycardia, bronchospasmserious

Brief — but contraindicated in asthma.

Flecainide pro-arrhythmiaserious

Increased mortality post-MI (CAST trial) — structural heart disease is the contraindication.

Lidocaine: CNS toxicity (perioral tingling, seizures)common

Cautions & contraindications

Adenosine in asthma/COPDasthma

Bronchospasm — use verapamil for SVT instead.

Flecainide in structural / ischaemic heart diseaseall

Pro-arrhythmic, ↑mortality.

AV-nodal blockers (adenosine/verapamil/digoxin) in AF with WPWall

Promote accessory-pathway conduction → VF.

Interactions

  • Dipyridamole potentiates adenosine; theophylline blocks it
  • Flecainide + AV-node blockers

Monitoring & kinetics

Continuous ECG during adenosine/IV antiarrhythmics

Adenosine IV push (seconds); flecainide oral; lidocaine/procainamide IV.

Source: Resus Council UK — Tachycardia · BNF — Antiarrhythmics