The drug atlas
Endocrine & Metabolic/Corticosteroid (glucocorticoid)

Corticosteroids (systemic)

also: prednisolone · hydrocortisone · dexamethasone · glucocorticoid · steroids

Overview

Cross-cutting anti-inflammatory/immunosuppressant used across nearly every specialty. The adverse-effect profile, the never-stop-abruptly rule and sick-day rules are core exam content.

Mechanism

Bind cytoplasmic glucocorticoid receptors → modulate gene transcription: ↓pro-inflammatory cytokines/COX-2/phospholipase A₂, suppressed immune-cell function (anti-inflammatory + immunosuppressive). Mineralocorticoid activity (esp. hydrocortisone) → Na⁺/water retention, K⁺ loss.

Indications

  • Inflammatory/autoimmune disease, asthma/COPD exacerbations, allergy/anaphylaxis (adjunct)
  • Replacement in adrenal insufficiency (hydrocortisone)
  • Croup, cerebral oedema, antenatal lung maturation (dexamethasone) — cross-references

The agents

Prednisoloneoral glucocorticoid

OD morning

Workhorse oral steroid.

Hydrocortisonegluco + mineralocorticoid

IV/oral

Acute (anaphylaxis, Addisonian crisis) + replacement.

Dexamethasonepotent, long-acting, no mineralocorticoid

Croup, cerebral oedema, antenatal, antiemetic.

Adverse effects

Cushingoid (moon face, central obesity, striae)classic
Hyperglycaemia / steroid-induced diabetesserious
Osteoporosisserious

Bone protection if long-term.

Immunosuppression / infection (incl. reactivation)serious
Adrenal suppression → Addisonian crisis if stopped abruptlyserious

Never stop long-term steroids suddenly — taper; sick-day rules (double dose when ill).

Peptic ulcer, mood/psychosis, proximal myopathy, cataracts/glaucoma, hypertension, hypokalaemiacommon

Cautions & contraindications

Systemic infection (relative)all
Live vaccines if significantly immunosuppressedall
Abrupt withdrawal after prolonged useall

Adrenal crisis.

Interactions

  • NSAIDs → GI ulcer
  • ↑glucose (antagonise antidiabetics)
  • CYP inducers reduce efficacy
  • Live vaccines

Monitoring & kinetics

Glucose, BP, weight; bone protection + PPI if long-term; growth in children,Steroid treatment card for >3 weeks

Oral/IV/IM/topical/inhaled. Give oral once daily in the morning (mimics circadian cortisol).

Source: BNF — Corticosteroids · NICE CKS — Corticosteroids