The drug atlas
Neurology/Stroke & acute neuro therapeutics

Stroke, GBS, MND & raised ICP drugs

also: alteplase thrombolysis · aspirin stroke · riluzole · IVIG Guillain-Barre · mannitol

Overview

The acute-neurology drug decisions — ischaemic stroke (thrombolysis/antiplatelets), Guillain-Barré, motor neurone disease, and raised intracranial pressure.

Mechanism

Alteplase (tPA) activates plasminogen → fibrinolysis (thrombolysis within 4.5 h, after haemorrhage excluded). Aspirin/clopidogrel are antiplatelets (secondary prevention). Riluzole inhibits glutamate release (modest survival benefit in MND). IVIG/plasma exchange remove pathogenic antibody (GBS). Dexamethasone reduces tumour-associated oedema; mannitol/hypertonic saline osmotically reduce ICP.

Indications

  • Acute ischaemic stroke / TIA
  • Guillain-Barré syndrome
  • Motor neurone disease
  • Raised ICP / cerebral oedema

The agents

Aspirin 300 mg → clopidogrelischaemic stroke

Aspirin 300 mg for 2 weeks after stroke (exclude bleed first), then clopidogrel long-term; AF → anticoagulate.

Alteplasethrombolysis

within 4.5 h

After CT excludes haemorrhage + no contraindications; ± thrombectomy.

IVIG / plasma exchangeGuillain-Barré

Steroids do NOT help GBS; monitor FVC (respiratory failure).

RiluzoleMND

Modest survival benefit; + NIV/nutrition.

Dexamethasone / mannitolraised ICP

Dexamethasone for tumour oedema; mannitol/hypertonic saline for acute ICP.

Adverse effects

Alteplase: intracranial/systemic haemorrhageserious
Antiplatelet bleedingcommon
Riluzole: hepatotoxicity (monitor LFTs)common

Cautions & contraindications

Thrombolysis with haemorrhage / recent surgery / bleeding / >4.5 hall

Catastrophic bleeding.

Steroids in Guillain-Barréall

Ineffective — use IVIG/PLEX.

Interactions

  • Thrombolysis + anticoagulants/antiplatelets ↑bleeding

Monitoring & kinetics

Stroke: CT before/after; GBS/MND: FVC; riluzole: LFTs

Time-critical (thrombolysis <4.5 h). See Antiplatelets/Anticoagulants cards (CV) for secondary prevention detail.

Source: NICE NG128 — Stroke/TIA · BNF — Stroke